Contents.- v.1 Global perspective, v.2 Strategy and drug research, v.3 Drug discovery technologies, v.4 Computer assisted drug design, v.5 ADME-Tox approaches, v.6 Therapeutic areas l : central nervous system, pain, metabolic syndrome, urology, gastrointestinal and cardiovascular, v.7 Therapeutic areas l : cancer, infectious disease, inflammation and immunology and dermatology, v.8 Case histories and cumulative subject index.